Cinolazepam

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Not to be confused with clonazepam or camazepam. ‹See Tfd›
Cinolazepam
Cinolazepam.svg
Cinolazepam3d.png
Systematic (IUPAC) name
(RS)-3-[9-Chloro-6-(2-fluorophenyl)-4-hydroxy-3-oxo-2,5-diazabicyclo[5.4.0]undeca-5,8,10,12-tetraen-2-yl]propanenitrile
Clinical data
AHFS/Drugs.com International Drug Names
Pregnancy cat. ?
Legal status Schedule IV (US)
Routes Oral
Pharmacokinetic data
Bioavailability 90-100%
Metabolism Hepatic
Half-life 9 h[1]
Excretion Renal
Identifiers
CAS number 75696-02-5 YesY
ATC code N05CD13
PubChem CID 3033621
DrugBank DB01594
ChemSpider 2298251 YesY
UNII 68P0556B0U YesY
KEGG D07328 YesY
ChEBI CHEBI:59514 YesY
ChEMBL CHEMBL2104926
Chemical data
Formula C18H13ClFN3O2 
Mol. mass 357.8
 YesY (what is this?)  (verify)

Cinolazepam[2] (marketed under the brand name Gerodorm)[3] is a drug which is a benzodiazepine derivative. It possesses anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties. Due to its strong sedative properties, it is primarily used as an hypnotic.

Cinolazepam is not approved for sale in the United States or Canada.

See also[edit]

References[edit]

  1. ^ Saletu, B.; G. Kindshofer; P. Anderer; J. Grunberger (1987). "Short-term sleep laboratory studies with cinolazepam in situational insomnia induced by traffic noise.". International Journal of Clinical Pharmacology Research 7 (5): 407–18. PMID 2889679. 
  2. ^ US Patent 4388313 Novel 3-hydroxy-1,4-benzodiazepine-2-ones and process for the preparation thereof
  3. ^ Lannacher Romania (1999). "Gerodorm". Produse Gerot inregistrate in Romania (in Romanian). Archived from the original on 11 October 2006. Retrieved 17 August 2006. 

External links[edit]