Pipamperone

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Pipamperone
Pipamperone1.svg
Systematic (IUPAC) name
1'-[4-(4-fluorophenyl)-4-oxobutyl]-1,4'-bipiperidine-4'-carboxamide
Clinical data
AHFS/Drugs.com International Drug Names
Oral
Identifiers
1893-33-0 N
N05AD05
PubChem CID 4830
IUPHAR ligand 92
ChemSpider 4664 YesY
UNII 5402501F0W YesY
KEGG D02622 YesY
ChEMBL CHEMBL440294 YesY
Chemical data
Formula C21H30FN3O2
375.480 g/mol
 N (what is this?)  (verify)

Pipamperone is an antipsychotic drug (a butyrophenone derivative) used in the treatment of schizophrenia. Pipamperone is known to the general public under the marketed brand name Dipiperon. It was discovered at Janssen Pharmaceutica in 1960.

Pipamperon neuraxpharm, 40mg

Synthesis[edit]

  • U.S. Patent 3,041,344
  • DE 1,235,319 
  • Van De Westeringh, C.; Van Daele, P.; Hermans, B.; Van Der Fycken, C.; Boey, J.; Janssen, P. A. J. (1964). "4-Substituted Piperidines. I. Derivatives of 4-t-Amino-4-piperidinecarboxamides". Journal of Medicinal Chemistry 7 (5): 619. doi:10.1021/jm00335a010.  edit

See also[edit]

References[edit]