Template:Antiarrhythmic agents
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Antiarrhythmic agents
(
C01B
)
Channel blockers
class I
(
Na
+
channel blockers
)
class Ia (
Phase 0
→ and
Phase 3
→)
Procainamide
#
Quinidine
#
Ajmaline
Disopyramide
Prajmaline
Lorajmine
Sparteine
class Ib (
Phase 3
←)
IV
(
Lidocaine
#)
enteral
(
Mexiletine
Tocainide
Aprindine
)
class Ic (
Phase 0
→)
Encainide
‡
Flecainide
Lorcainide
Moracizine
‡
Propafenone
class III
(
Phase 3
→,
K
+
channel blockers
)
Amiodarone
Dronedarone
Bretylium
Bunaftine
Dofetilide
Ibutilide
Nifekalant
Sotalol
Tedisamil
Vernakalant
E-4031
class IV
(
Phase 4
→,
Ca
2+
channel blockers
)
Verapamil
#
Diltiazem
Receptor
agonists
and
antagonists
class II
(
Phase 4
→,
β blockers
)
Propranolol
Nadolol
Pindolol
cardioselective
(
Atenolol
Metoprolol
Acebutolol
Esmolol
)
A1 agonist
Adenosine
M2
muscarinic antagonist
:
Atropine
Quinidine
Disopyramide
muscarinic agonist
:
Digoxin
α receptors
Quinidine
Verapamil
Amiodarone
Bretylium
Ion transporters
Na
+
/ K
+
-ATPase
Digoxin
#
WHO-EM
‡
Withdrawn
from market
Clinical trials
:
†
Phase III
§
Never to phase III
M
:
HRT
anat
/
phys
/
devp
noco
/
cong
/
tumr
,
sysi
/
epon
,
injr
proc
,
drug
(
C1A
/
1B
/
1C
/
1D
),
blte
Categories
:
Antiarrhythmic agents
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