Valperinol

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Valperinol
Valperinol.svg
Systematic (IUPAC) name
(1R,3R,4S,6R,7S,8R,10R)-8-methoxy-10-methyl-3-(1-piperidinylmethyl)-2,9-dioxatricyclo[4.3.1.03,7]decan-4-ol
Clinical data
Legal status Non-regulated
Identifiers
CAS number 64860-67-9
ATC code None
PubChem CID 68849
ChemSpider 62082
Chemical data
Formula C16H27NO4 
Mol. mass 297.390 g/mol

Valperinol (INN; GA 30-905) is a drug which acts as a calcium channel blocker.[1][2] It was patented as a possible sedative, antiepileptic, and/or antiparkinsonian agent, but was never marketed.[3]

References[edit]

  1. ^ Thies PW, Asai A, Bán I, David S, Finner E (1984). "[The synthesis of valperinol and various 3-aminomethyl derivatives of 2,9-dioxatricyclo[4,3,1,0(3,7)]decane from didrovaltrate]". Arzneimittel-Forschung (in German) 34 (11): 1460–3. PMID 6543120. 
  2. ^ Dose M (1984). "[Calcium antagonist properties of valperinol]". Arzneimittel-Forschung (in German) 34 (11): 1464–6. PMID 6098282. 
  3. ^ Dictionary of Pharmacological Agents Volume 2. CRC Press. p. 2104. ISBN 978-0-412-46630-4. Retrieved 22 April 2012.