BzODZ-EPyr is an indole based synthetic cannabinoid that has been sold as a designer drug in Russia.
It acts as a CB1 receptor agonist with a pKB value of 7.2 and demonstrates that replacing the ketone in 3-carbonylindoles with an oxadiazole spacer does generally not lead to activity loss.
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- ^ Moloney, Peter Gerard; Robertson, Alan Duncan (2005), "Patent US6930118 - 3-Oxadiazol-5-yl-1-aminoalkyl-1h-indole derivatives", Amrad Operations Pty. Ltd.