CUMYL-PINACA

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CUMYL-PINACA
CUMYL-PINACA.png
Legal status
Legal status
Identifiers
CAS Number
PubChem CID
ChemSpider
Chemical and physical data
Formula C22H27N3O
Molar mass 349.5 g/mol
3D model (JSmol)

CUMYL-PINACA (also known as SGT-24) is an indazole-3-carboxamide based synthetic cannabinoid. CUMYL-PINACA acts as a potent agonist for the cannabinoid receptors, with approximately 3x selectivity for CB1, having an EC50 of 0.15nM for human CB1 receptors and 0.41nM for human CB2 receptors.[1] In its pure form, it is described as a sticky oil which can cause poisoning through transdermal exposure.[2]

Legal status[edit]

Sweden's public health agency suggested to classify CUMYL-PINACA as hazardous substance on November 10, 2014.[3]

See also[edit]

References[edit]

  1. ^ Bowden; et al. (11 April 2013). "Patent WO 2014167530 - Cannabinoid compounds". New Zealand Patent application 623626. Retrieved 11 July 2015. 
  2. ^ Dobaja M, Grenc D, Kozelj G, Brvar M. Occupational transdermal poisoning with synthetic cannabinoid cumyl-PINACA. Clin Toxicol. 2017 Mar;55(3):193-195. doi: 10.1080/15563650.2016.1278224. PMID 28084855
  3. ^ "Cannabinoider föreslås bli klassade som hälsofarlig vara". Retrieved 11 July 2015.