Ethyl carfluzepate

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Ethyl carfluzepate
Ethyl carfluzepate.svg
Identifiers
CAS Number
PubChem CID
ChemSpider
UNII
Chemical and physical data
Formula C20H17ClFN3O4
Molar mass 417.818
3D model (Jmol)
 NYesY (what is this?)  (verify)

Ethyl carfluzepate[1] is mainly a hypnotic drug which is a benzodiazepine derivative and induces sleep in a strong manner. It is similar to ethyl loflazepate in chemical structure, the other difference being an absence of methylcarbamoyl group. Its also similar in metabolism to this substance, only the methyl-carboxylate group would be the difference between the main metabolites. Two of the main metabolites must be the 3-hydroxylate or the substance with only a hydrogen atom at the 3-position of the molecule structure. In order to that the resulting main metabolite could probably be ethyl-7-cloro-5-(2-fluorophenyl)-1-methylcarbamate)-2-oxo-3H-1,4-benzodiazepine-3-hydroxylate (and the 3-OH instead of the 3H metabolite). Its properties are mainly sedative and hypnotic.[2][3]

References[edit]

  1. ^ DE 2719607 
  2. ^ "ethyl carfluzepate". psychotropics.dk. 2003. Retrieved 7 December 2009. 
  3. ^ "LIST OF INTERNATIONAL NON-PROPRIETARY NAMES (INNS), PROVIDED FOR PHARMACEUTICAL SUBSTANCES BY THE WORLD HEALTH ORGANIZATION, WHICH ARE FREE OF DUTY" (PDF). Official Journal of the European Communities. eur-lex.europa.eu. 23 October 2001. Retrieved 7 December 2009.