Exaprolol

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Exaprolol
Exaprolol.svg
Names
IUPAC name
1-(2-Cyclohexylphenoxy)-3-(propan-2-ylamino)propan-2-ol
Other names
Esprolol
Identifiers
Jmol interactive 3D Image
PubChem 65485
Properties
C18H29NO2
Molar mass 291.44 g·mol−1
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
Infobox references

Exaprolol is a beta-adrenoceptor antagonist.[1]

Synthesis[edit]

Exaprolol synthesis:[2]

References[edit]

  1. ^ Van Waarde, A; Doorduin, J; De Jong, JR; Dierckx, RA; Elsinga, PH (2008). "Synthesis and preliminary evaluation of (S)-11C-exaprolol, a novel beta-adrenoceptor ligand for PET". Neurochemistry international 52 (4–5): 729–33. doi:10.1016/j.neuint.2007.09.009. PMID 17961850. 
  2. ^ Carissimi, M; Gentili, P; Grumelli, E; Milla, E; Picciola, G; Ravenna, F (1976). "Basic ethers of cyclohexylphenols with beta-blocking activity: Synthesis and pharmacological study of exaprolol". Arzneimittel-Forschung 26 (4): 506–16. PMID 8056.