List of opioids

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Opium poppy (Papaver somniferum) flower

This is a list of opioids, opioid antagonists and inverse agonists.

Opium and poppy straw derivatives[edit]

Seedhead of opium poppy with white latex

Crude opiate extracts whole opium products[edit]

Natural opiates[edit]

Opium alkaloids[edit]

Alkaloid salts mixtures[edit]

Semisynthetics including Bentley compounds[edit]

Morphine family[edit]

3,6-diesters of morphine[edit]

Codeine-dionine family[edit]

Morphinones and morphols[edit]

Morphides[edit]

Dihydrocodeine series[edit]

Nitrogen morphine derivatives[edit]

Hydrazones[edit]

Halogenated morphine derivatives[edit]

Active opiate metabolites[edit]

Morphinans[edit]

Morphinan series[edit]

Others[edit]

Benzomorphans[edit]

4-Phenylpiperidines[edit]

Pethidines (meperidines)[edit]

Prodines[edit]

Ketobemidones[edit]

Others[edit]

Open chain opioids[edit]

Amidones[edit]

Methadols[edit]

Moramides[edit]

Thiambutenes[edit]

Phenalkoxams[edit]

Ampromides[edit]

Others[edit]

Anilidopiperidines[edit]

Oripavine derivatives[edit]

Thienorphine

Phenazepanes[edit]

Pirinitramides[edit]

Benzimidazoles[edit]

Indoles[edit]

Beta-Amino Ketones[edit]

Diphenylmethylpiperazines[edit]

Opioid peptides[edit]

Dynorphins[edit]

Endomorphins[edit]

Endorphins[edit]

Enkephalins[edit]

Propeptides[edit]

Others / unknown[edit]

Others[edit]

Opioid antagonists and inverse agonists[edit]

Biased ligands[edit]

Receptor heteromer targeting ligands[edit]

Uncategorized opioids[edit]

Combination drug formulations containing opioids[edit]

See also[edit]

References[edit]

  1. ^ ChemIndex CAS Registry Number 3371-56-0
  2. ^ ChemIndex CAS Registry Number 509-56-8
  3. ^ ChemIndex CAS Registry Number 63715-94-6
  4. ^ NCBI PubChem SID 750205
  5. ^ chembase cbid_346222
  6. ^ Gomes I, Fujita W, Gupta A, Saldanha SA, Saldanha AS, Negri A, Pinello CE, Eberhart C, Roberts E, Filizola M, Hodder P, Devi LA (2013). "Identification of a μ-δ opioid receptor heteromer-biased agonist with antinociceptive activity". Proc. Natl. Acad. Sci. U.S.A. 110 (29): 12072–7. doi:10.1073/pnas.1222044110. PMC 3718106. PMID 23818586. 
  7. ^ Yekkirala AS, Lunzer MM, McCurdy CR, Powers MD, Kalyuzhny AE, Roerig SC, Portoghese PS (2011). "N-naphthoyl-beta-naltrexamine (NNTA), a highly selective and potent activator of μ/kappa-opioid heteromers". Proc. Natl. Acad. Sci. U.S.A. 108 (12): 5098–103. doi:10.1073/pnas.1016277108. PMC 3064379. PMID 21385944. 

External links[edit]

  • Carbonate derivatives of 14β-hydroxycodeine "viz., 14β-hydroxy-6-O-(methoxycarbonyl)codeine, 6-O-methoxycarbonyl-14β-(methoxycarbonyloxy)codeine, and 14β-acetoxy-6-O-methoxy-carbonylcodeine, potential substrates for ring C modification in morphinane (sic) alkaloids, were synthesized for the first time." Russian Chemical Bulletin. August 2008, Volume 57, Issue 8, pp 1773–1774. Date: 11 Aug 2009; I. V. Evsikova, S. K. Moiseev, P. V. Petrovskii, V. N. Kalinin. Published in Russian in Izvestiya Akademii Nauk. Seriya Khimicheskaya, No. 8, pp. 1739–1740