SB-200646

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SB-200646
SB-200646.svg
Clinical data
ATC code
  • none
Legal status
Legal status
  • UN: Unscheduled
Identifiers
PubChem CID
ChemSpider
KEGG
ChEBI
ChEMBL
Chemical and physical data
Formula C15H14N4O
Molar mass 302.76 g/mol
3D model (JSmol)

SB-200646 is a 5-HT2 receptor antagonist with anxiolytic properties in rats. It was the first 5-HT2 antagonist discovered to have selectivity of 5-HT2C/2B over 5-HT2A.[1]

References[edit]

  1. ^ Kennett, GA; Wood, MD; Glen, A; Grewal, S; Forbes, I; Gadre, A; Blackburn, TP (1994), "In vivo properties of SB 200646A, a 5-HT2C/2B receptor antagonist", Br J Pharmacol, British Journal of Pharmacology, 111: 797–802, doi:10.1111/j.1476-5381.1994.tb14808.x, PMC 1910094Freely accessible, PMID 7912626