Search results
The page "Bisubstrate+analogue" does not exist. You can create a draft and submit it for review or request that a redirect be created, but consider checking the search results below to see whether the topic is already covered.
(August 1996). "2.3 A resolution X-ray crystal structure of the bisubstrate analogue inhibitor salicylhydroxamic acid bound to human myeloperoxidase:...17 KB (1,879 words) - 23:40, 27 April 2024
catalytic center of ATCase was first made possible by the binding of a bisubstrate analogue, N-(phosphonoacetyl)-L-aspartate (PALA). This compound is a strong...18 KB (2,141 words) - 08:46, 4 May 2024
N-acetylserotonin. Based on this mechanism, it might be expected that a bisubstrate analog inhibitor, derived from the tethering of indole and CoASH parts...25 KB (2,982 words) - 13:11, 26 August 2023
enzymology with previously utilized inhibition motifs. For example, a "bisubstrate analog" inhibits kinase action by binding both the conserved ATP binding...55 KB (6,090 words) - 01:19, 20 March 2024
"Catechol-O-methyltransferase in complex with substituted 3'-deoxyribose bisubstrate inhibitors". Acta Crystallographica. Section D, Biological Crystallography...22 KB (2,140 words) - 01:13, 9 March 2024
N1-acetyltransferase superinduced in response to treatment with antitumor polyamine analogues". Cancer Research. 54 (15): 3955–8. PMID 8033120. Xiao L, Casero RA (January...18 KB (2,126 words) - 17:52, 9 January 2024
Ward SG (April 2010). "Toward the development of potent and selective bisubstrate inhibitors of protein arginine methyltransferases". Bioorganic & Medicinal...111 KB (12,530 words) - 17:53, 14 April 2024
- products. Sequential reactions can be either ordered or random. In a bisubstrate reaction, a ternary complex of the enzyme and both substrates forms.