Template:Neuromodulation
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Neuromodulation
Types
♦
Enzyme
:
Inducer
Inhibitor
♦
Ion channel
:
Opener
Blocker
♦
Receptor
:
Agonist
Antagonist
Positive allosteric modulator
(PAM)
Negative allosteric modulator
(NAM)
Inverse agonist
♦
Transporter
[
Reuptake
]:
Enhancer
(RE)
Inhibitor
(RI)
Releaser
(RA)
♦ Miscellaneous:
Precursor
Cofactor
Classes
Enzyme
see
Enzyme inhibition
Ion channel
Calcium channel blocker
(CCB)
Potassium channel blocker
(PCB)
Sodium channel blocker
(SCB)
Potassium channel opener
(PCO)
Receptor
&
transporter
BA
/
M
Adrenergic
Adrenergic receptor agonist
(
α
β
(
1
2
))
Adrenergic receptor antagonist
(
α
(
1
2
),
β
)
Adrenergic reuptake inhibitor
(ARI)
Dopaminergic
Dopamine receptor agonist
Dopamine receptor antagonist
Dopamine reuptake inhibitor
(DRI)
Histaminergic
Histamine receptor agonist
Histamine receptor antagonist
(
H
1
H
2
H
3
)
Serotonergic
Serotonin receptor agonist
Serotonin Receptor Antagonist
(
5-HT
3
)
Serotonin reuptake inhibitor
(SRI)
Serotonin reuptake enhancer
(SRE)
AA
GABAergic
GABA receptor agonist
GABA receptor antagonist
GABA reuptake inhibitor
(GRI)
Glutamatergic
Glutamate receptor agonist
(
AMPA
)
Glutamate receptor antagonist
(
NMDA
)
Cholinergic
Acetylcholine receptor agonist
(
Muscarinic
Nicotinic
)
Acetylcholine receptor antagonist
(
Muscarinic
Nicotinic
(
Ganglionic
Muscular
))
Endocannabinoid
Cannabinoid receptor agonist
Cannabinoid receptor antagonist
Opioid
Opioid receptor agonist
Opioid receptor antagonist
Other
Adenosine reuptake inhibitor
(AdoRI)
Angiotensin II receptor antagonist
Endothelin receptor antagonist
NK
1
receptor antagonist
Vasopressin receptor antagonist
Miscellaneous
Cofactor
(see
Enzyme cofactors
)
Precursor
(see
Amino acids
)
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