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MDMA (redirect from Ecstacy (drug))Guillon JM (2014). "Safety Pharmacology assessment of drugs with biased 5-HT(2B) receptor agonism mediating cardiac valvulopathy". Journal of Pharmacological...166 KB (15,881 words) - 07:54, 15 August 2024
Agonist (redirect from Receptor agonism)Terms that describe this phenomenon are "functional selectivity", "protean agonism", or selective receptor modulators. As mentioned above, agonists have the...14 KB (1,622 words) - 03:21, 4 September 2024
Aripiprazole (category Drugs with non-standard legal status)D2-dopamine receptors are clearly cell-type specific (e.g., agonism, antagonism, partial agonism), and are most parsimoniously explained by the "functional...105 KB (9,662 words) - 17:36, 29 August 2024- Anxiolytic (redirect from Antianxiety drug)MT1 receptor agonism, MT3 receptor antagonism, and sigma receptor agonism thought to have some involvement. Bromantane is a stimulant drug with anxiolytic...46 KB (4,436 words) - 22:29, 27 August 2024
5-MeO-DiPT (redirect from Foxy (drug))effects of 5-MeO-DiPT is thought to result primarily from 5-HT2A receptor agonism, although additional mechanisms of action such as monoamine oxidase inhibition...9 KB (719 words) - 16:47, 2 September 2024
both a tryptamine and lysergamide). They act via serotonin 2A receptor agonism. When compounds bind to serotonin 5-HT2A receptors, they modulate the activity...83 KB (8,663 words) - 00:10, 4 September 2024
Fabomotizole (category Drugs missing an ATC code)GABAergic, NGF- and BDNF-release-promoting, MT1 receptor agonism, MT3 receptor antagonism, and sigma agonism suggested as potential mechanisms. Fabomotizole was...6 KB (453 words) - 11:30, 4 June 2024- Efficacy (redirect from Drug effect)by the conformation change from shut to open. It was found that partial agonism results from deficiency in the first step, and that the opening and shutting...13 KB (1,523 words) - 22:13, 27 February 2024
- Synthetic drugs refer to substances that are artificially modified from naturally-occurring drugs and are capable of exhibiting both therapeutic and psychoactive...25 KB (2,877 words) - 22:38, 8 December 2023
Antibody–drug conjugates or ADCs are a class of biopharmaceutical drugs designed as a targeted therapy for treating cancer. Unlike chemotherapy, ADCs are...41 KB (4,305 words) - 11:56, 24 August 2024
Methaqualone (redirect from Lemmon (drug))transmission and downstream sedative effects via allosteric modulation and agonism of several GABAAR subtypes. Similar to other GABAergic agents, methaqualone...25 KB (2,518 words) - 00:21, 31 August 2024
and potent agonists of the trace amine-associated receptor 1 (TAAR1); agonism of TAAR1 triggers phosphorylation events that result in both non-competitive...6 KB (418 words) - 04:31, 25 July 2024- Functional selectivity (redirect from Biased agonism)Functional selectivity (or “agonist trafficking”, “biased agonism”, “biased signaling”, "ligand bias" and “differential engagement”) is the ligand-dependent...17 KB (1,848 words) - 23:24, 8 July 2024
Tirzepatide (category Drugs with non-standard legal status)receptor and distinct signaling properties at GLP-1 suggest this biased agonism increases insulin secretion. Tirzepatide has been reported to increase...44 KB (3,528 words) - 18:08, 3 September 2024
mechanism that evolved to help increase the adaptive fitness of animals. In drug addiction, certain substances over-activate the reward circuit, leading to...103 KB (12,754 words) - 12:31, 2 September 2024
5-MeO-MiPT (category Chemical pages without DrugBank identifier)effects of 5-MeO-MiPT is thought to result primarily from 5-HT2A receptor agonism, although additional mechanisms of action such as inhibition of MAO may...12 KB (1,038 words) - 05:51, 8 June 2024
Cocaine (redirect from Coke (drug))Smith SL (December 2014). "Dopamine reuptake transporter (DAT) "inverse agonism"--a novel hypothesis to explain the enigmatic pharmacology of cocaine"...177 KB (18,939 words) - 13:25, 31 August 2024
Receptor antagonist (redirect from Antagonist drug)at high or low levels. In addition, it has been suggested that partial agonism prevents the adaptive regulatory mechanisms that frequently develop after...33 KB (3,845 words) - 01:47, 19 August 2024- GLP-1 receptor agonist (redirect from GLP-1 drug)the amount of weight loss caused by the drugs. Combination with glucagon agonism is likely to make the drugs more efficacious for weight loss, at the...37 KB (3,890 words) - 03:08, 12 August 2024
Antihistamine (redirect from Anti-histamine drug)R, Church MK, Taglialatela M (April 2002). "H1-antihistamines: inverse agonism, anti-inflammatory actions and cardiac effects". Clinical and Experimental...32 KB (3,140 words) - 11:09, 17 August 2024
- warm the soul Bright Helen mix'd a mirth-inspiring bowl, Temper'd with drugs, of sovereign use t'assuage The boiling bosom of tumultuous rage; To clear
- ferocious anachronisms: nuclear jihad in the Indian subcontinent; the medieval agonism of Islam; the Bronze Age blunderings of the Middle East. … The champions
- Antineoplastic drugs are drugs that are used to eliminate patient's neoplastic processes. Neoplasms are types of abnormal and excessive growths, called