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Quinaprilat Other names CI-928 ATC code
(3S )-2-[(2S )-2-[[(1S )-1-carboxy-3-phenylpropyl]amino]propanoyl]-3,4-dihydro-1H -isoquinoline-3-carboxylic acid
CAS Number IUPHAR/BPS ChemSpider UNII ChEMBL CompTox Dashboard (EPA ) Formula C 23 H 26 N 2 O 5 Molar mass 410.46294 g·mol−1 3D model (JSmol )
C[C@@H](C(=O)N1CC2=CC=CC=C2C[C@H]1C(=O)O)N[C@@H](CCC3=CC=CC=C3)C(=O)O
InChI=1S/C23H26N2O5/c1-15(24-19(22(27)28)12-11-16-7-3-2-4-8-16)21(26)25-14-18-10-6-5-9-17(18)13-20(25)23(29)30/h2-10,15,19-20,24H,11-14H2,1H3,(H,27,28)(H,29,30)/t15-,19-,20-/m0/s1
Key:FLSLEGPOVLMJMN-YSSFQJQWSA-N
Quinaprilat is the active metabolite of quinapril .[ 1]
References
^ Ferry, J J; Horvath, A M; Sedman, A J; Latts, J R; Colburn, W A (1987). "Influence of food on the pharmacokinetics of quinapril and its active diacid metabolite, CI-928". Journal of clinical pharmacology . 27 (5): 397–399. doi :10.1002/j.1552-4604.1987.tb03037.x .
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