Terbequinil

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Terbequinil
Terbequinil structure.png
Systematic (IUPAC) name
1-(methoxymethyl)-4-oxo-N-propylquinoline-3-carboxamide
Clinical data
Legal status
?
Identifiers
CAS number 113079-82-6
ATC code None
PubChem CID 65916
ChemSpider 59325 YesY
UNII 0DH9WUS03O YesY
Chemical data
Formula C15H18N2O3 
Mol. mass 274.315 g/mol
 YesY (what is this?)  (verify)

Terbequinil (SR-25776) is a stimulant and nootropic drug which acts as a partial inverse agonist at benzodiazepine sites on the GABAA receptor. In human trials it was found to partially reverse the sedative and amnestic effects of the hypnotic drug triazolam with only slight effects when administered by itself.[1]

See also[edit]

References[edit]

  1. ^ Warot D, Danjou P, Douillet P, Keane P, Puech AJ. Cognitive impairments induced by triazolam in healthy volunteers: antagonism by a partial inverse agonist of benzodiazepine receptor. Therapie. 1994 Jan-Feb;49(1):23-6. PMID 8091361