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{{Drugbox
| Verifiedfields = changed
| Watchedfields = changed
| verifiedrevid = 457138752
| IUPAC_name = 4-[(1R )-1-hydroxy-2-{[4-(4-hydroxyphenyl)butyl]amino}ethyl]benzene-1,2-diol
| image = Arbutamine.svg
| width = 250
| tradename =
| pregnancy_AU =
| pregnancy_US =
| pregnancy_category =
| legal_AU =
| legal_CA =
| legal_UK =
| legal_US =
| legal_status =
| routes_of_administration =
| bioavailability =
| protein_bound =
| metabolism =
| elimination_half-life =
| excretion =
| CAS_number_Ref = Y
| CAS_number = 128470-16-6
| ATC_prefix = C01
| ATC_suffix = CA22
| PubChem = 60789
| DrugBank_Ref = Y
| DrugBank = DB01102
| ChemSpiderID_Ref = Y
| ChemSpiderID = 54785
| UNII_Ref = Y
| UNII = B07L15YAEV
| ChEBI_Ref = Y
| ChEBI = 50580
| ChEMBL_Ref = N
| ChEMBL = 1201251
| C=18 | H=23 | N=1 | O=4
| molecular_weight = 317.38 g/mol
| smiles = Oc1ccc(cc1O)[C@@H](O)CNCCCCc2ccc(O)cc2
| StdInChI_Ref = Y
| StdInChI = 1S/C18H23NO4/c20-15-7-4-13(5-8-15)3-1-2-10-19-12-18(23)14-6-9-16(21)17(22)11-14/h4-9,11,18-23H,1-3,10,12H2/t18-/m0/s1
| StdInChIKey_Ref = Y
| StdInChIKey = IIRWWTKISYTTBL-SFHVURJKSA-N
}}
Arbutamine is a cardiac stimulant . It stimulates β adrenergic receptors .[ 1]
References
^ Abou-Mohamed, Gamal; Nagarajan, Ravi; Ibrahim, Tarek M.; Caldwell, Robert W. (March 1996). "Characterization of the Adrenergic Activity of Arbutamine, a Novel Agent for Pharmacological Stress Testing". Cardiovascular Drugs and Therapy . 10 (1): 39–47. doi :10.1007/BF00051129 . PMID 8723169 .
α1
Agonists Antagonists
Abanoquil Ajmalicine Alfuzosin Anisodamine Anisodine Atiprosin Atypical antipsychotics (e.g., brexpiprazole , clozapine , olanzapine , quetiapine , risperidone )Benoxathian Beta blockers (e.g., adimolol , amosulalol , arotinolol , carvedilol , eugenodilol , labetalol )Buflomedil Bunazosin Corynanthine Dapiprazole Domesticine Doxazosin Ergolines (e.g., acetergamine , ergotamine , dihydroergotamine , lisuride , nicergoline , terguride )Etoperidone Fenspiride Hydroxyzine Indoramin Ketanserin L-765,314 mCPP Mepiprazole Metazosin Monatepil Moxisylyte Naftopidil Nantenine Neldazosin Niaprazine Niguldipine Pardoprunox Pelanserin Perlapine Phendioxan Phenoxybenzamine Phentolamine Phenylpiperazine antidepressants (e.g., hydroxynefazodone , nefazodone , trazodone , triazoledione )Piperoxan Prazosin Quinazosin Quinidine Silodosin Spegatrine Spiperone Talipexole Tamsulosin Terazosin Tiodazosin Tolazoline Tetracyclic antidepressants (e.g., amoxapine , maprotiline , mianserin )Tricyclic antidepressants (e.g., amitriptyline , clomipramine , doxepin , imipramine , trimipramine )Trimazosin Typical antipsychotics (e.g., chlorpromazine , fluphenazine , loxapine , thioridazine )Urapidil WB-4101 Zolertine
α2
Agonists Antagonists
1-PP Adimolol Amesergide Aptazapine Atipamezole Atypical antipsychotics (e.g., asenapine , brexpiprazole , clozapine , lurasidone , olanzapine , paliperidone , quetiapine , risperidone , zotepine )Azapirones (e.g., buspirone , gepirone , ipsapirone , tandospirone )BRL-44408 Buflomedil Cirazoline Efaroxan Esmirtazapine Fenmetozole Fluparoxan Idazoxan Ketanserin Lisuride mCPP Mianserin Mirtazapine NAN-190 Pardoprunox Phentolamine Phenoxybenzamine Piperoxan Piribedil Rauwolscine Rotigotine Setiptiline Spegatrine Spiroxatrine Sunepitron Terguride Tolazoline Typical antipsychotics (e.g., chlorpromazine , fluphenazine , loxapine , thioridazine )Yohimbine
β
| CAS_number = 128470-16-6
| ATC_prefix = C01
| ATC_suffix = CA22
| PubChem = 60789
| DrugBank_Ref = 
| ChEMBL = 1201251
