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Arformoterol Trade names Brovana AHFS /Drugs.com Monograph MedlinePlus a602023 License data
Routes of administration Inhalation solution for nebuliser ATC code Legal status
Protein binding 52–65% Elimination half-life 26 hours
N -[2-hydroxy-5-[(1R )-1-hydroxy-2-[[(2R )-1-(4-methoxyphenyl) propan-2-yl]amino]ethyl] phenyl]formamide
CAS Number PubChem CID IUPHAR/BPS DrugBank ChemSpider UNII ChEBI ChEMBL CompTox Dashboard (EPA ) Formula C 19 H 24 N 2 O 4 Molar mass 344.405 g/mol g·mol−1
InChI=1S/C19H24N2O4/c1-13(9-14-3-6-16(25-2)7-4-14)20-11-19(24)15-5-8-18(23)17(10-15)21-12-22/h3-8,10,12-13,19-20,23-24H,9,11H2,1-2H3,(H,21,22)/t13-,19+/m1/s1
Y Key:BPZSYCZIITTYBL-YJYMSZOUSA-N
Y
N Y (what is this?) (verify)
Arformoterol is a long-acting β2 adrenoreceptor agonist (LABA) indicated for the treatment of chronic obstructive pulmonary disease (COPD). It is sold by Sunovion , under the trade name Brovana , as a solution of arformoterol tartrate to be administered twice daily (morning and evening) by nebulization .[1]
It is the active (R ,R )-(−)-enantiomer of formoterol and was approved by the United States Food and Drug Administration (FDA) on October 6, 2006 for the treatment of COPD.
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