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==References==
==References==
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{{reflist}}

{{Opioids}}

[[Category:Opioids]]


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Revision as of 19:49, 19 October 2012

14-Ethoxymetopon
Clinical data
Other names14-Ethoxymetopon
Identifiers
  • 3-hydroxy- 14-ethoxy- 5-methyl- 7,8-dihydro- 4,5α-epoxy- 17-methylmorphinan- 6-one
CAS Number
PubChem CID
ChemSpider
CompTox Dashboard (EPA)
Chemical and physical data
FormulaC20H25NO4
Molar mass343.42 g/mol g·mol−1
3D model (JSmol)
  • CCOC12CCC(=O)[C@@]3(C14CCN([C@@H]2CC5=C4C(=C(C=C5)O)O3)C)C
  • InChI=1S/C20H25NO4/c1-4-24-20-8-7-15(23)18(2)19(20)9-10-21(3)14(20)11-12-5-6-13(22)17(25-18)16(12)19/h5-6,14,22H,4,7-11H2,1-3H3/t14-,18-,19?,20?/m1/s1 checkY
  • Key:LDTUYTORBPKTNO-HPJZBDCMSA-N checkY
 ☒NcheckY (what is this?)  (verify)

14-Ethoxymetopon[1] is an opiate analogue that is a derivative of metopon which has been substituted with an ethoxy group at the 14-position. It is a highly potent analgesic drug several hundred times stronger than morphine.[2]

References

  1. ^ US Patent 6476044
  2. ^ Fürst, Z; Búzás, B; Friedmann, T; Schmidhammer, H; Borsodi, A (1993). "Highly potent novel opioid receptor agonist in the 14-alkoxymetopon series". European Journal of Pharmacology. 236 (2): 209–15. doi:10.1016/0014-2999(93)90591-5. PMID 8391457.