Binaltorphimine

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Binaltorphimine
Binaltorphimine.svg
Clinical data
ATC code
  • None
Identifiers
CAS Number
PubChem CID
ChemSpider
ChEMBL
Chemical and physical data
Formula C41H45N3O6
Molar mass 675.813 g/mol
3D model (JSmol)

Binaltorphimine (BNI) is a selective antagonist of the κ-opioid receptor (KOR).[1] BNI and norbinaltorphimine (nor-BNI) were the first highly selective KOR antagonists to be discovered.[1]

See also[edit]

References[edit]

  1. ^ a b Portoghese PS, Lipkowski AW, Takemori AE (March 1987). "Binaltorphimine and nor-binaltorphimine, potent and selective kappa-opioid receptor antagonists". Life Sci. 40 (13): 1287–92. PMID 2882399. doi:10.1016/0024-3205(87)90585-6.