Opioid modulator
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This is an old revision of this page, as edited by Ffffrr (talk | contribs) at 08:55, 16 April 2022 (Adding short description: "Drug" (Shortdesc helper)). The present address (URL) is a permanent link to this revision, which may differ significantly from the current revision.
Revision as of 08:55, 16 April 2022 by Ffffrr (talk | contribs) (Adding short description: "Drug" (Shortdesc helper))
Drug
An opioid modulator (or opioid receptor modulator) is a drug which has mixed agonist and antagonist actions at different opioid receptors and thus cannot clearly be described as either an opioid agonist or antagonist. An example of an opioid modulator is buprenorphine, which is a partial agonist of the μ-opioid receptor and an antagonist of the κ-opioid receptor.[1]
See also
References
- ^ Hillemacher T, Heberlein A, Muschler MA, Bleich S, Frieling H (August 2011). "Opioid modulators for alcohol dependence". Expert Opin Investig Drugs. 20 (8): 1073–86. doi:10.1517/13543784.2011.592139. PMID 21651459.