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Piperidylthiambutene

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Piperidylthiambutene
Clinical data
ATC code
  • none
Identifiers
  • 1-[4,4-Di(thiophen-2-yl)but-3-en-2-yl]piperidine
CAS Number
PubChem CID
ChemSpider
CompTox Dashboard (EPA)
Chemical and physical data
FormulaC17H21NS2
Molar mass303.485 g/mol g·mol−1
3D model (JSmol)
Melting point188 to 189 °C (370 to 372 °F)
  • C1CCCCN1C(C)C=C(c3cccs3)c2sccc2
  • InChI=1S/C17H21NS2/c1-14(18-9-3-2-4-10-18)13-15(16-7-5-11-19-16)17-8-6-12-20-17/h5-8,11-14H,2-4,9-10H2,1H3
  • Key:FQRWJLVMJCKSME-UHFFFAOYSA-N
  (verify)

Piperidylthiambutene (Piperidinohton) is an opioid analgesic drug from the thiambutene family, which has around the same potency as morphine.[1][2][3] If sold / was obtained for the purpose of human consumption it could be considered a controlled substance analogue in some countries such as the USA, Australia and New Zealand, but is legal in the rest of the world.

References

  1. ^ Adamson DW, Green AF. A new series of analgesics. Nature. 1950 Jan 21;165(4186):122. doi:10.1038/165122a0 PMID 15409854
  2. ^ Adamson DW, Duffin WM, Green AF. Dithienylbutylamines as analgesics. Nature. 1951 Jan 27;167(4239):153-4. doi:10.1038/167153b0 PMID 14806409
  3. ^ Green AF. Analgesic and other properties of 3: 3-dithienylalkenylamines. British Journal of Pharmacology and Chemotherapy. 1953 Mar;8(1):2-9. PMID 13066683