Avitriptan

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Avitriptan
Avitriptan.png
Systematic (IUPAC) name
1-[3-[3-[4-(5-methoxypyrimidin-4-yl)piperazin-1-yl]propyl]-1H-indol-5-yl]-N-methyl-methanesulfonamide
Clinical data
Legal status
?
Identifiers
CAS number 151140-96-4 N
ATC code None
PubChem CID 133081
ChemSpider 117442 YesY
UNII 6RS056L04P YesY
ChEMBL CHEMBL2105880 N
Chemical data
Formula C22H30N6O3S 
Mol. mass 458.58 g/mol
 N (what is this?)  (verify)

Avitriptan (INN) (code name BMS-180,048) is an antimigraine drug of the triptan family which was never marketed.[1] It acts as a 5-HT1B and 5-HT1D receptor agonist.[1]

See also[edit]

References[edit]

  1. ^ a b Saxena PR, De Vries P, Wang W, et al. (February 1997). "Effects of avitriptan, a new 5-HT 1B/1D receptor agonist, in experimental models predictive of antimigraine activity and coronary side-effect potential". Naunyn-Schmiedeberg's Archives of Pharmacology 355 (2): 295–302. doi:10.1007/pl00004946. PMID 9050026.