Trestolone enanthate
This is an old revision of this page, as edited by Citation bot (talk | contribs) at 19:34, 7 September 2020 (Alter: pages. Add: s2cid. Formatted dashes. | You can use this bot yourself. Report bugs here. | Suggested by Abductive | Category:Abandoned drugs | via #UCB_Category). The present address (URL) is a permanent link to this revision, which may differ significantly from the current revision.
Clinical data | |
---|---|
Other names | Trestolone 17β-enanthate; MENT enanthate; 7α-Methyl-19-nortestosterone 17β-enanthate; 7α-Methylestr-4-en-17β-ol-3-one 17β-enanthate |
Pregnancy category |
|
Drug class | Androgen; Anabolic steroid; Androgen ester |
Identifiers | |
| |
CAS Number | |
Chemical and physical data | |
Formula | C26H40O3 |
Molar mass | 400.603 g·mol−1 |
3D model (JSmol) | |
| |
|
Trestolone enanthate, also known as 7α-methyl-19-nortestosterone 17β-enanthate (MENT enanthate), is an androgen and anabolic steroid (AAS) and progestogen which was never marketed.[1][2] It is an androgen ester; specifically, it is the C17β enanthate (heptanoate) ester of trestolone (7α-methylestr-4-en-17β-ol-3-one).[2] Trestolone enanthate has low affinity for sex hormone-binding globulin (SHBG), similarly to testosterone enanthate.[1]
See also
References
- ^ a b Cunningham GR, Tindall DJ, Lobl TJ, Campbell JA, Means AR (September 1981). "Steroid structural requirements for high affinity binding to human sex steroid binding protein (SBP)". Steroids. 38 (3): 243–62. doi:10.1016/0039-128X(81)90061-1. PMID 7197818. S2CID 2702353.
- ^ a b Bursi R, Grootenhuis A, van der Louw J, Verhagen J, de Gooyer M, Jacobs P, Leysen D (March 2003). "Structure-activity relationship study of human liver microsomes-catalyzed hydrolysis rate of ester prodrugs of MENT by comparative molecular field analysis (CoMFA)". Steroids. 68 (3): 213–220. doi:10.1016/S0039-128X(02)00186-1. PMID 12628684. S2CID 32309966.
ERTooltip Estrogen receptor |
| ||||||
---|---|---|---|---|---|---|---|
GPERTooltip G protein-coupled estrogen receptor |
| ||||||
PRTooltip Progesterone receptor |
| ||||||
---|---|---|---|---|---|---|---|
mPRTooltip Membrane progesterone receptor (PAQRTooltip Progestin and adipoQ receptor) |
| ||||||
This drug article relating to the genito-urinary system is a stub. You can help Wikipedia by expanding it. |
- Articles with short description
- Short description is different from Wikidata
- Drugs with non-standard pregnancy category
- Articles without EBI source
- Chemical pages without ChemSpiderID
- Chemical pages without DrugBank identifier
- Articles without KEGG source
- Articles without UNII source
- Drugs missing an ATC code
- Drugs with no legal status
- Articles containing unverified chemical infoboxes
- All stub articles